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Albiglutide information


Albiglutide
Clinical data
Trade namesEperzan (Europe), Tanzeum (US)
Other namesGSK-716155
AHFS/Drugs.comtanzeum
Routes of
administration
Subcutaneous (SC)
ATC code
  • A10BJ04 (WHO)
Legal status
Legal status
  • CA: ℞-only[1]
  • US: ℞-only
Pharmacokinetic data
Protein bindingProbably none
MetabolismMost likely proteolysis
Elimination half-life5 (4–7) days
Identifiers
CAS Number
  • 782500-75-8
PubChem SID
  • 96025526
DrugBank
  • DB09043
ChemSpider
  • none
UNII
  • 5E7U48495E
KEGG
  • D08843
Chemical and physical data
FormulaC3232H5032N864O979S41
Molar mass72971.34 g·mol−1

Albiglutide (trade names Eperzan in Europe and Tanzeum in the US) is a glucagon-like peptide-1 agonist (GLP-1 agonist) drug marketed by GlaxoSmithKline (GSK) for treatment of type 2 diabetes. As of 2017 it is unclear if it affects a person's risk of death.[2] GSK has announced that it intends to withdraw the drug from the worldwide market by July 2018 for economic reasons.

  1. ^ "Health Canada New Drug Authorizations: 2015 Highlights". Health Canada. 4 May 2016. Retrieved 7 April 2024.
  2. ^ Liu J, Li L, Deng K, Xu C, Busse JW, Vandvik PO, et al. (June 2017). "Incretin based treatments and mortality in patients with type 2 diabetes: systematic review and meta-analysis". BMJ. 357: j2499. doi:10.1136/bmj.j2499. PMC 5463186. PMID 28596247.

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