The adenosine A2A receptor, also known as ADORA2A, is an adenosine receptor, and also denotes the human gene encoding it.[5][6]
^ abcGRCh38: Ensembl release 89: ENSG00000128271 – Ensembl, May 2017
^ abcGRCm38: Ensembl release 89: ENSMUSG00000020178 – Ensembl, May 2017
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^"Mouse PubMed Reference:". National Center for Biotechnology Information, U.S. National Library of Medicine.
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four known types of adenosinereceptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene. The adenosinereceptors are commonly known...
Cellular signaling by adenosine occurs through four known adenosinereceptor subtypes (A1, A2A, A2B, and A3). Extracellular adenosine concentrations from...
The adenosine A1 receptor (A1AR) is one member of the adenosinereceptor group of G protein-coupled receptors with adenosine as endogenous ligand. A1 receptors...
subtypes of adenosine A2 receptors are known. Both are G protein-coupled adenosinereceptors: AdenosineA2AreceptorAdenosine A2B receptor This disambiguation...
receptors on the neutrophil, and the affinity of these receptors for adenosine. Micromolar concentrations of adenosine activate A2A and A2B receptors...
enkephalin and a high density of dopamine D2 and adenosineA2Areceptors (they also express adenosine A1 receptors), while dynorphinergic MSNs connect the striatum...
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The adenosine A3 receptor, also known as ADORA3, is an adenosinereceptor, but also denotes the human gene encoding it. Adenosine A3 receptors are G protein-coupled...
agonist. A2AR & A2BR: The AdenosineA2Areceptor is regarded as an important checkpoint in cancer therapy because adenosine in the immune microenvironment...
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one adenosine A1 receptor and one dopamine D1 receptor) and the A2A–D2 receptor heterotetramer (this is a receptor complex with two adenosineA2A receptors...
(specifically, the medium spiny neurons of the D2-type which co-express adenosineA2Areceptors), and a GABAergic nucleus in the lateral hypothalamus which co-releases...
The adenosine A2B receptor, also known as ADORA2B, is a G-protein coupled adenosinereceptor, and also denotes the human adenosine A2b receptor gene which...
Therapeutics for an undisclosed sum, as well as licensing PBF-509, an adenosineA2Areceptor antagonist which is in Phase I clinical trials for non-small cell...
Schering-Plough which acted as a potent and selective antagonist at the adenosineA2Areceptor. It was being researched as a potential treatment for Parkinson's...
P2Y receptors are a family of purinergic G protein-coupled receptors, stimulated by nucleotides such as adenosine triphosphate, adenosine diphosphate...
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