Histamine agonist information

A histamine agonist is a drug which causes increased activity at one or more of the four histamine receptor subtypes. H2: Betazole and Impromidine are...

inverse agonist at histamine receptors. Only a few currently marketed H1-antihistamines are known to function as inverse agonists. Histamine makes blood vessels...

affecting their activity. The drug betazole is an example of a histamine H2 receptor agonist. Histamine is a ubiquitous messenger molecule released from mast cells...

histamine receptor belonging to the family of rhodopsin-like G-protein-coupled receptors. This receptor is activated by the biogenic amine histamine....

selectivity; partial agonist effects on cAMP inhibition and MAPK activity, antagonist on histamine release, and inverse agonist on arachidonic acid release)...

H1-antihistamines. Virtually all H1-antihistamines function as inverse agonists at the histamine H1-receptor, as opposed to neutral antagonists, as was previously...

at histamine H3 receptors and a weak agonist at histamine H1 receptors. Betahistine has two mechanisms of action. Primarily, it is a weak agonist at histamine...

Histamine is an organic nitrogenous compound involved in local immune responses communication, as well as regulating physiological functions in the gut...

Parasympathomimetic drug (acetylcholine agonist) Histamine agonist Borovac JA (March 2016). "Side effects of a dopamine agonist therapy for Parkinson's disease: a mini-review...

efficacy. Receptors for which inverse agonists have been identified include the GABAA, melanocortin, mu opioid, histamine and beta adrenergic receptors. Both...

The histamine H4 receptor, like the other three histamine receptors, is a member of the G protein-coupled receptor superfamily that in humans is encoded...

Methimepip is a histamine agonist which is highly selective for the H3 subtype. It is the N-methyl derivative of immepip. Kitbunnadaj R, Hashimoto T,...

and histamine H1 receptor. Lisuride is a partial agonist of the D2, D3, D4, 5-HT2A, 5-HT2C, 5-HT5A, and H1 receptors, a full or near-full agonist of the...

histamine H3 receptor ligand which is a "protean agonist", producing different effects ranging from full agonist, to antagonist, to inverse agonist in...

Ciproxifan is an extremely potent histamine H3 inverse agonist/antagonist. The histamine H3 receptor is an inhibitory autoreceptor located on histaminergic...

inhibitor (NDRI), and pitolisant, which acts as a histamine 3 (H3) receptor antagonist/inverse agonist. Cephalon, the original U.S. market rights holder...

physiological agonists to each other. There are several substances that have antihistaminergic action despite not being ligands for the histamine receptor...

A GABA receptor agonist is a drug that is an agonist for one or more of the GABA receptors, producing typically sedative effects, and may also cause other...

potent and specific histamine H2 receptor agonist. It has been used diagnostically as a gastric secretion indicator. Histamine agonists Durant G, Duncan...

Histamine trifluoromethyl toluidide (HTFMT) is a mixed H1/H2 histamine agonist which is significantly more potent than histamine itself. It also produces...

the agonist histamine which contains an imidazole ring in its structure. The structural diversity among H3R is limited and all known H3R agonists today...

blockers, are a class of medications that block the action of histamine at the histamine H2 receptors of the parietal cells in the stomach. This decreases...