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Valerylfentanyl information


Valerylfentanyl
Legal status
Legal status
  • BR: Class F1 (Prohibited narcotics)
  • CA: Schedule I
  • DE: Anlage II (Authorized trade only, not prescriptible)
  • UK: Class A
  • US: Schedule I
  • UN: Narcotic Schedule I
Identifiers
IUPAC name
  • N-(1-(2-Phenylethyl)-4-piperidinyl)-N-phenylpentylamide
CAS Number
  • 122882-90-0
PubChem CID
  • 21595398
ChemSpider
  • 10551383
UNII
  • VUG0EQK700
KEGG
  • C22762
CompTox Dashboard (EPA)
  • DTXSID801014173 Edit this at Wikidata
Chemical and physical data
FormulaC24H32N2O
Molar mass364.533 g·mol−1
3D model (JSmol)
  • Interactive image
SMILES
  • CCCCC(=O)N(C1CCN(CC1)CCC2=CC=CC=C2)C3=CC=CC=C3
InChI
  • InChI=1S/C24H32N2O/c1-2-3-14-24(27)26(22-12-8-5-9-13-22)23-16-19-25(20-17-23)18-15-21-10-6-4-7-11-21/h4-13,23H,2-3,14-20H2,1H3
  • Key:VCCPXHWAJYWQMR-UHFFFAOYSA-N

Valerylfentanyl is an opioid analgesic that is an analog of fentanyl and has been sold online as a designer drug.[1] It has been seldom reported on illicit markets and there is little information about it, though it is believed to be less potent than butyrfentanyl but more potent than benzylfentanyl.[2] In one study, it fully substituted for oxycodone and produced antinociception and oxycodone-like discriminative stimulus effects comparable in potency to morphine in mice,[3] but failed to stimulate locomotor activity in mice at doses up to 100 mg/kg.[4]

  1. ^ Cooman T, Hoover B, Sauvé B, Bergeron SA, Quinete N, Gardinali P, Arroyo LE (June 2022). "The metabolism of valerylfentanyl using human liver microsomes and zebrafish larvae". Drug Testing and Analysis. 14 (6): 1116–1129. doi:10.1002/dta.3233. PMID 35128825. S2CID 246633284.
  2. ^ Prekupec MP, Mansky PA, Baumann MH (2017). "Misuse of Novel Synthetic Opioids: A Deadly New Trend". Journal of Addiction Medicine. 11 (4): 256–265. doi:10.1097/ADM.0000000000000324. PMC 5537029. PMID 28590391.
  3. ^ Walentiny DM, Moisa LT, Beardsley PM (May 2019). "Oxycodone-like discriminative stimulus effects of fentanyl-related emerging drugs of abuse in mice". Neuropharmacology. 150: 210–216. doi:10.1016/j.neuropharm.2019.02.007. PMID 30735691.
  4. ^ Varshneya NB, Walentiny DM, Moisa LT, Walker TD, Akinfiresoye LR, Beardsley PM (June 2019). "Opioid-like antinociceptive and locomotor effects of emerging fentanyl-related substances". Neuropharmacology. 151: 171–179. doi:10.1016/j.neuropharm.2019.03.023. PMC 8992608. PMID 30904478. S2CID 84182661.

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