Fentanyl azepane (Fentanyl azepane homologue) is an opioid derivative which is a homologue of fentanyl, where the central piperidine ring has been expanded to an azepane ring. It is many times less potent than fentanyl itself, being only slightly stronger than morphine, but is still more potent than the ring-contracted pyrrolidine derivative, as well as other related compounds such as benzylfentanyl and ethoheptazine. The β-hydroxy derivative is slightly more potent again, as with betahydroxyfentanyl.[1][2][3]
^Deruiter J, Andurkar S, Riley TN, Walters DE, Noggle Jr FT (1992). "Investigation of the synthesis and analgesic activity of 1-substituted 4-(propananilido) perhydroazepines". Journal of Heterocyclic Chemistry. 29 (4): 779–786. doi:10.1002/jhet.5570290417.
^Vardanyan RS, Hruby VJ (March 2014). "Fentanyl-related compounds and derivatives: current status and future prospects for pharmaceutical applications". Future Medicinal Chemistry. 6 (4): 385–412. doi:10.4155/fmc.13.215. PMC 4137794. PMID 24635521.
Fentanylazepane (Fentanylazepane homologue) is an opioid derivative which is a homologue of fentanyl, where the central piperidine ring has been expanded...
This is a list of fentanyl analogues (sometimes referred to as Fentalogs), including both compounds developed by pharmaceutical companies for legitimate...
weaker, only around the same potency as morphine. Fentanylazepane Secofentanyl Phenaridine List of fentanyl analogues Riley TN, Bagley JR (October 1979)....
Butyrylfentanyl Fentanylazepane Isofentanyl Secofentanyl OPPPP Cooper D, Jacob M, Allen A (April 1986). "Identification of fentanyl derivatives". Journal...
synthetic cannabinoids Arylcyclohexylamines List of aminorex analogues List of fentanyl analogues List of methylphenidate analogues Meltzer PC, Butler D, Deschamps...
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