Norethisterone acetate, a widely used progestogen ester and prodrug of norethisterone.Medroxyprogesterone acetate, a progestogen ester that does not act as a prodrug.
This is a list of progestogen esters, or esters of progestogens.[1][2][3][4]
Unlike the case of testosterone and estradiol, progesterone cannot be esterified as it lacks hydroxyl groups, so all progestogen esters, with the exception of esters of 17α-hydroxyprogesterone like hydroxyprogesterone caproate, are esters of progestins (synthetic progestogens) and are non-bioidentical. In addition, whereas all androgen and estrogen esters are prodrugs of the parent compound, only some and not all progestogen esters act as prodrugs. Esters of 17α-hydroxyprogesterone and 19-norprogesterone derivatives like hydroxyprogesterone caproate, medroxyprogesterone acetate, and nomegestrol acetate are active themselves and are not prodrugs, whereas esters of 19-nortestosterone derivatives like norethisterone acetate and norethisterone enanthate are not active themselves and are prodrugs.
^J. Elks (14 November 2014). The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. ISBN 978-1-4757-2085-3.
^Index Nominum 2000: International Drug Directory. Taylor & Francis. January 2000. ISBN 978-3-88763-075-1.
^"List of Progestins".
^Sweetman, Sean C., ed. (2009). "Sex hormones and their modulators". Martindale: The Complete Drug Reference (36th ed.). London: Pharmaceutical Press. ISBN 978-0-85369-840-1.
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A progestogenester is an esterof a progestogen or progestin (a synthetic progestogen). The prototypical progestogen is progesterone, an endogenous sex...
This is a listof androgen esters, including esters (as well as ethers) of natural androgens like testosterone and dihydrotestosterone (DHT) and synthetic...
group of progestins. Note that although an active progestogen, SC-5233 (spirolactone) is not medically used. Listof steroids Listofprogestogenesters ?...
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This is a listofprogestogens (progesterone and progestins) and formulations that are approved by the FDATooltip Food and Drug Administration in the United...
replacement therapy (ART), among other indications. Examples of androgen esters include testosterone esters such as testosterone cypionate, testosterone enanthate...
enanthate, is a form of hormonal birth control which is used to prevent pregnancy in women. It is used both as a form ofprogestogen-only injectable birth...
(methylsuperlutin), which is used in veterinary medicine. Listofprogestogenesters § Estersof 17α-hydroxyprogesterone derivatives 16-Methylene-17α-hydroxyprogesterone...
caproate, megestrol caproate, and methenmadinone caproate. Listofprogestogenesters § Estersof 17α-hydroxyprogesterone derivatives Daniel R. Mishell (1983)...
powerlifters. Side effects of nandrolone esters include masculinization among others. In women, nandrolone and nandrolone esters have been reported to produce increased...
Estrogen-progestogen Menopausal Therapy. World Health Organization. pp. 417–. ISBN 978-92-832-1291-1. Norethisterone and its acetate and enanthate esters are...
intrauterine device (IUD), also known as an intrauterine system (IUS) with progestogen and sold under the brand name Mirena among others, is an intrauterine...
progestin, or a synthetic progestogen, and hence is an agonist of the progesterone receptor, the biological target ofprogestogens like progesterone. The...
SAAs also act as potent progestogens and therefore antigonadotropins. Note that this list does not include pure progestogens, only SAAs also acting as...
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